Publications of the Synthetic Chemistry Group

2017


Massai, D., Bolesani, E., Robles Diaz, D., Kropp, C., Kempf, H., Halloin, C., Martin, U., Braniste, T., Isu, G., Harms, V., Morbiducci, U., Dräger, G., & Zweigerdt, R. (2017). Sensitivity of human pluripotent stem cells to insulin precipitation induced by peristaltic pump-based medium circulation: Considerations on process development. Scientific Reports, 7(1), Article 3950. https://doi.org/10.1038/s41598-017-04158-x
Ringel, M. T., Dräger, G., & Brüser, T. (2017). The periplasmic transaminase PtaA of Pseudomonas fluorescens converts the glutamic acid residue at the pyoverdine fluorophore to α-ketoglutaric acid. Journal of Biological Chemistry, 292(45), 18660-18671. https://doi.org/10.1074/jbc.M117.812545
Ammermann, J., Schmidt, T., Donner, J., Reck, M., Dalton, M., Stumpp, N., Stiesch, M., Wagner-Döbler, I., & Kirschning, A. (2017). The carolactam strategy is ineffective: synthesis and biological evaluation of carolactam. Organic and Biomolecular Chemistry, 15(40), 8553-8558. https://doi.org/10.1039/c7ob02060k
Mohammadi-Ostad-Kalayeh, S., Hrupins, V., Helmsen, S., Ahlbrecht, C., Stahl, F., Scheper, T., Preller, M., Surup, F., Stadler, M., Kirschning, A., & Zeilinger, C. (2017). Development of a microarray-based assay for efficient testing of new HSP70/DnaK inhibitors. Bioorganic and Medicinal Chemistry, 25(24), 6345-6352. https://doi.org/10.1016/j.bmc.2017.10.003
Seidel, K., Balakrishnan, A., Alexiou, C., Janko, C., Komoll, R. M., Wang, L., Kirschning, A., & Ott, M. (2017). Synthesis of Magnetic-Nanoparticle/Ansamitocin Conjugates: Inductive Heating Leads to Decreased Cell Proliferation In Vitro and Attenuation Of Tumour Growth In Vivo. Chemistry - A European Journal, 23(50), 12326-12337. https://doi.org/10.1002/chem.201701491
Donner, J., Reck, M., Bunk, B., Jarek, M., App, C. B., Meier-Kolthoff, J. P., Overmann, J., Müller, R., Kirschning, A., & Wagner-Döbler, I. (2017). The biofilm inhibitor carolacton enters Gram-negative cells: Studies using a Tol-Cdeficient strain of Escherichia coli. mSphere, 2(5), Article e00375-17. https://doi.org/10.1128/mspheredirect.00375-17
Wang, L., Candito, D., Dräger, G., & Kirschning, A. (2017). Synthetic Studies Probing Elansolid Biosynthesis: A para-Quinone-Methide-Triggered Intramolecular Diels–Alder Reaction. European Journal of Organic Chemistry, 2017(37), 5582-5591. https://doi.org/10.1002/ejoc.201701125
Sommer, H., Braun, M., Schröder, B., & Kirschning, A. (2017). 4-Ethoxy-1,1,1-trifluoro-3-buten-2-one (ETFBO), a Versatile Precursor for Trifluoromethyl-Substituted Heteroarenes: A Short Synthesis of Celebrex ® (Celecoxib). Synlett, 29(1), 121-125. Article st-2017-b0101-l. https://doi.org/10.1055/s-0036-1589097
Kirschning, A., Dibbert, N., & Dräger, G. (2017). Chemical Functionalization of Polysaccharides: Towards Biocompatible Hydrogels for Biomedical Applications. Chemistry - A European Journal, 24(6), 1231-1240. https://doi.org/10.1002/chem.201701906
Hüttel, S., Testolin, G., Herrmann, J., Planke, T., Gille, F., Moreno, M., Stadler, M., Brönstrup, M., Kirschning, A., & Müller, R. (2017). Discovery and Total Synthesis of Natural Cystobactamid Derivatives with Superior Activity against Gram-Negative Pathogens. Angewandte Chemie , 56(41), 12760-12764. https://doi.org/10.1002/anie.201705913, https://doi.org/10.1002/ange.201705913