Publications

Journale

  • Attique Ahmed, Pervaiz Ali Channar, Aamer Saeed, Markus Kalesse, Mehar Ali Kazi, Fayaz Ali Larik, Qamar Abbas, Mubashir Hassan, Hussain Raza, Sung-Yum Seo (2019) Synthesis of sulfonamide, amide and amine hybrid pharmacophore, an entry of new class of carbonic anhydrase II inhibitors and evaluation of chemo-informatics and binding analysisBioorganic Chemistry 2019, 86, 624
    DOI: 10.1016/j.bioorg.2019.01.060
  • Dr. Jørn Eivind Tungen, Dr. Lisa Gerstmann, Prof. Dr. Anders Vik, Roberta De Matteis, Dr. Romain, Alexandre Colas, Prof. Dr. Jesmond Dalli, Prof. Dr. Nan Chiang, Prof. Dr. Charles Nicholas Serhan, Prof. Dr. Markus Kalesse, Prof. Dr. Trond Vidar Hansen (2019) Resolving Inflammation: Synthesis, Configurational Assignment, and Biological Evaluations of RvD1n−3 DPAChem. Eur. J. 2019, 25, 1476 –1480
    DOI: 10.1002/chem.201806029
  • Luebken, D.; Saxarra, M.; Kalesse, M. (2019) Tris(acetylacetonato) Iron (III): Recent Developments and Synthetic Applications.Synthesis-Stuttgart, 2019, 51(1), 161-177
    DOI: 10.1055/s-0037-1610393
  • Claudia Brandt,. Patricia Seja, Kathrin Töllner, Kerstin Römermann, Philip Hampel, Markus Kalesse, Andi Kipper, Peter W. Feit, Kasper Lykke, Trine Lisberg Toft-Bertelsen, Pauliina Paavilainen, Inkeri Spoljaric, Martin Puskarjov, Nanna MacAulaye, Kai Kaila, Wolfgang Löscher (2018) Bumepamine, a brain-permeant benzylamine derivative of bumetanide, does not inhibit NKCC1 but is more potent to enhance phenobarbital's anti-seizure efficacyNeuropharmacology, 2018, 143, 186-204
    DOI: 10.1016/j.neuropharm.2018.09.025
  • Li, J.; Xing, J.; Luecke, D.; Luebken, D.; Millbrodt, L.; Plentz, R. R.; Kalesse, M. (2018) The Structure Elucidation of Haprolid.Synthesis-Stuttgart 2018, 50(3), 529-538
    DOI: 10.1055/s-0036-1591836
  • Luecke, D.; Linne, Y.; Hempel, K.; Kalesse, M. (2018) Total Synthesis of Pericoannosin A.Organic Letters 2018, 20(15), 4475-4477
    DOI: 10.1021/acs.orglett.8b01768
  • Stempel, E.; Kaml, R. F.-X.; Budisa, N.; Kalesse, M. (2018) Painting argyrins blue: Negishi cross-coupling for synthesis of deep-blue tryptophan analogue beta-(1-azulenyl)-L-alanine and its incorporation into argyrin C.Bioorgan. Med. Chem. 2018, 26(19), 5259-5269
    DOI: 10.1016/j.bmc.2018.03.037
  • Surup, F.; Kuhnert, E.; Boehm, A.; Pendzialek, T.; Solga, D.; Wiebach, V.; Engler, H.; Berkessel, A.; Stadler, M.; Kalesse, M. (2018) The Rickiols: 20-, 22-, and 24-membered Macrolides from the Ascomycete Hypoxylon rickii.Chem-Eur. J. 2018, 24(9), 2200-2213
    DOI: 10.1002/chem.201704928
  • A. Feklistov, B. Bae, J. Hauver, A. Lass-Napiorkowska, M. Kalesse, F. Glaus, K.-H. Altmann, T. Heyduk, R. Landick, S. A. Darst (2017) RNA polymerase motions during promoter meltingScience, 2017, 356, 863
    DOI: 10.1126/science.aam7858
  • B. Werner, M. Kalesse (2017) Pinacol Coupling Strategy for the Construction of the Bicyclo[6.4.1]tridecane Framework of Schiglautone AOrg. Lett., 2017, 19, 1524
    DOI: 10.1021/acs.orglett.7b00288
  • Poock, C.; Kalesse, M. (2017) Total Synthesis of Nannocystin Ax.Organic Letters 2017, 19(17), 4536-4539
    DOI: 10.1021/acs.orglett.7b02112
  • Witte, S. N. R.; Hug, J. J.; Geraldy, M. N. E.; Mueller, R.; Kalesse, M. (2017) Biosynthesis and Total Synthesis of Pyrronazol B: a Secondary Metabolite from Nannocystis pusilla.Chem. Eur. J. 2017, 23(63), 15917-15921
    DOI: 10.1002/chem.201703782
  • X. Chen, K. C. Bui, S. Barat, M. L. Thi Nguyen, P. Bozko, B. Sipos, M. Kalesse, N. P. Maleka, R. R. Plentz (2017) Therapeutic effects of Argyrin F in pancreatic adenocarcinomaCancer Lett., 2017, 399, 20
    DOI: 10.1016/j.canlet.2017.04.003
  • G. Parthasarathy, U. Eggert, M. Kalesse (2016) Synthesis of (+)-Omphadiol and (+)-Pyxidatol COrg. Lett., 2016, 18, 2320
    DOI: 10.1021/acs.orglett.6b00814
  • Gerstmann, L.; Kalesse, M. (2016) Total Synthesis of Aetheramide A.Chem-Eur. J. 2016, 22(32), 11210-11212
    DOI: 10.1002/chem.201602682
  • H. Steinmetz, J. Li, C. Fu, N. Zaburannyi, B. Kunze, K. Harmrolfs, V. Schmitt, J. Herrmann, H. Reichenbach, G. Höfle, M. Kalesse, R. Müller (2016) Isolation, Structure Elucidation, and (Bio)Synthesis of Haprolid, a Cell-Type-Specific Myxobacterial CytotoxinAngew. Chem. Int. Ed. 2016, 55, 10113
    DOI: 10.1002/anie.201603288
  • Steinmetz, H.; Li, J.; Fu, C.; Zaburannyi, N.; Kunze, B.; Harmrolfs, K.; Schmitt, V.; Herrmann, J.; Reichenbach, H.; Hoefle, G.; Kalesse, M.; Müller, R. (2016) Isolation, Structure Elucidation, and(Bio)Synthesis of Haprolid, a Cell-Type-Specific Myxobacterial Cytotoxin.Angew. Chem. Int. Edit. 2016, 55(34), 10113-10117
    DOI: 10.1002/anie.201603288
  • T. Tautz, J. Hoffmann, T. Hoffmann, H. Steinmetz, P. Washausen, B. Kunze, V. Huch, A. Kitsche, H. Reichenbach, G. Höfle, R. Müller, M. Kalesse (2016) Isolation, Structure Elucidation, Biosynthesis, and Synthesis of Antalid, a Secondary Metabolite from Polyangium speciesOrg. Lett., 2016, 18, 2560
    DOI: 10.1021/acs.orglett.6b00810
  • A. Naini, J. Fohrer, M. Kalesse (2015) The Synthesis of Desepoxy-Isotedanolide – A Potential Biosynthetic Precursor of TedanolideEur. J. Org. Chem. 2015, 4400
    DOI: 10.1002/ejoc.201500568
  • A. Naini, Y. Muthukumar, A. Raja, R. Franke, I. Harrier, A. B. Smith III, D. Lee, R. E. Taylor, F. Sasse, M. Kalesse (2015) The Synthesis and Biological Evaluation of Desepoxyisotedanolide and a Comparison with DesepoxytedanolideAngew. Chem. Int. Ed. 2015, 54, 6935
    DOI: 10.1002/anie.201501526
  • Bluhm, N.; Kalesse, M. (2015) Synthesis of a C20-Deoxygenated Spirangien Derivative for Target Identification.Synlett 2015, 26(6), 797-801
    DOI: 10.1055/s-0034-1379980
  • G. Koutsoudakis, I. Romero-Brey, C. Berger, G. Pérez-Vilaró, P. Monteiro Perin, F. W. R. Vondran, M. Kalesse, K. Harmrolfs, R. Müller, J. P. Martinez, T. Pietschmann, R. Bartenschlager, M. Brönstrup, A. Meyerhans, J. Díez (2015) Soraphen A: A broad-spectrum antiviral natural product with potent anti-hepatitis C virus activityJ. Hepatol. 2015, 63, 813
    DOI: 10.1016/j.jhep.2015.06.002
  • H.-H. Lu, B. Hinkelmann, T. Tautz, J. Li, F. Sasse, R. Franke, M. Kalesse (2015) Paleo-soraphens: chemical total syntheses and biological studiesOrg. Biomol. Chem. 2015, 13, 8029
    DOI: 10.1039/C5OB01249J
  • Lu, H.-H.; Hinkelmann, B.; Tautz, T.; Li, J.; Sasse, F.; Franke, R.; Kalesse, M. (2015) Paleo-soraphens: chemical total syntheses and biological studies.Org. Biomol. Chem. 2015, 13(29), 8029-8036
    DOI: 10.1039/c5ob01249j
  • M. Kalesse (2015) Ekkehard Winterfeldt (1932-2014)Angew. Chem. Int. Ed. 2015, 54, 35
    DOI: 10.1002/anie.201410838
  • N. Bluhm, M. Kalesse (2015) Synthesis of a C20-Deoxygenated Spirangien Derivative for Target IdentificationSynlett 2015, 26, 797
    DOI: 10.1055/s-0034-1379980
  • N. Bruns, W. Collisi, S. Bernecker, M. Stadler, C. Richter, H. Schwalbe, M. Kalesse (2015) Spirangien Derivatives from the Myxobacterium Sorangium cellulosum: Isolation, Structure Elucidation, and Biological ActivityEur. J. Org. Chem. 2015, 847
    DOI: 10.1002/ejoc.201403353
  • Naini, A.; Fohrer, J.; Kalesse, M. (2015) The Synthesis of Desepoxy-Isotedanolide - A Potential Biosynthetic Precursor of Tedanolide.Eur. J. Org. Chem. 2015, 20, 4400-4411
    DOI: 10.1002/ejoc.201500568
  • Naini, A.; Muthukumar, Y.; Raja, A.; Franke, R.; Harrier, I.; Smith, A. B., III; Lee, D.; Taylor, R. E.; Sasse, F.; Kalesse, M. (2015) The Synthesis and Biological Evaluation of Desepoxyisotedanolide and a Comparison with Desepoxytedanolide.Angew. Chem. Int. Edit. 2015, 54(23), 6935-6939
    DOI: 10.1002/anie.201501526
  • Gieseler, M. T.; Kalesse, M. (2014) Synthesis of Angiolam A.Organic Letters 2014, 16(2), 548-551
    DOI: 10.1021/ol403423r
  • H.-H. Lu, A. Raja, R. Franke, D. Landsberg, F. Sasse, M. Kalesse (2014) Synthesis and Biological Evaluation of Paleo-SoraphensAngew. Chem. Int. Ed. 2013, 52, 13549
    DOI: 10.1002/anie.201305331
  • Hartmann, O.; Kalesse, M. (2014) The Structure Elucidation and Total Synthesis of beta-Lipomycin.Angew. Chem. Int. Edit. 2014, 53(28), 7335-7338
    DOI: 10.1002/anie.201402259
  • J. Held, T. Gebru, M. Kalesse, R. Jansen, K. Gerth, R. Müller, B. Mordmüller (2014) Antimalarial Activity of the Myxobacterial Macrolide Chlorotonil AAntimicrob. Agents Chemother. 2014, 58, 6378
    DOI: 10.1128/AAC.03326-14
  • J. Niggemann, P. Bozko, N. Bruns, A. Wodtke, M. T. Gieseler, K. Thomas, C. Jahns, M. Nimtz, I. Reupke, T. Brüser, G. Auling, N. Malek, M. Kalesse (2014) Baceridin, a Cyclic Hexapeptide from an Epiphytic Bacillus Strain, Inhibits the ProteasomeChemBioChem 2014, 15, 1021
    DOI: 10.1002/cbic.201300778
  • Kalesse, M.; Cordes, M.; Symkenberg, G.; Lu, H.-H. (2014) The vinylogous Mukaiyama aldol reaction(VMAR) in natural product synthesis.Nat. Prod. Rep. 2014, 31(4), 563-594
    DOI: 10.1039/c3np70102f
  • Symkenberg, G.; Kalesse, M. (2014) Structure Elucidation and Total Synthesis of Kulkenon.Angew. Chem. Int. Edit. 2014, 53(7), 1795-1798
    DOI: 10.1002/anie.201309386
  • A. Kitsche, M. Kalesse (2013) Configurational Assignment of Secondary Hydroxyl Groups and Methyl Branches in Polyketide Natural Products through Bioinformatic Analysis of the Ketoreductase DomainChemBioChem 2013, 14, 851
    DOI: 10.1002/cbic.201300063
  • A. Rentsch, D. Landsberg, T. Brodmann, Tobias; L. Bülow, A.-K. Girbig, M. Kalesse (2013) Synthesis and Pharmacology of Proteasome InhibitorsAngew. Chem. Int. Ed. 2013, 52, 5450
    DOI: 10.1002/anie.201207900
  • D. Landsberg, O. Hartmann, U. Eggert, M. Kalesse (2013) Diastereodivergent Vinylogous Mukaiyama Aldol ReactionSynlett 2013, 1105
    DOI: 10.1055/s-0033-1338933
  • E. M. Borst, J. Kleine-Albers, I. Gabaev, M. Babic, K. Wagner, A. Binz, I. Degenhardt, M. Kalesse, S. Jonjic, R. Bauerfeind, M. Messerle (2013) The Human Cytomegalovirus UL51 Protein Is Essential for Viral Genome Cleavage-Packaging and Interacts with the Terminase Subunits pUL56 and pUL89J. Virol. 2013, 87, 1720
    DOI: 10.1128/JVI.01955-12
  • A. Rentsch, M. Kalesse (2012) The Total Synthesis of Corallopyronin A and Myxopyronin BAngew. Chem. 2012, 125, 11543
    DOI: 10.1002/anie.201206560
  • C. Jahns, T. Hoffmann, S. Müller, K. Gerth, P. Washausen, G. Höfle, H. Reichenbach, M. Kalesse, R. Müller (2012) Pellasoren: Structure Elucidation, Biosynthesis, and Total Synthesis of a Cytotoxic Secondary Metabolite from Sorangium cellulosumAngew. Chem. Int. Ed. 2012, 51, 5239
    DOI: 10.1002/anie.201200327
  • G. Symkenberg, M. Kalesse (2012) Syn-Selective Vinylogous Kobayashi Aldol ReactionOrg. Lett. 2012, 14, 1608
    DOI: 10.1021/ol300353w
  • M. Kalesse (2012) Biomimetic Organic Synthesis. Edited by Erwan Poupon and Bastien NayAngew. Chem. Int. Ed. 2012, 51, 583
    DOI: 10.1002/anie.201107291
  • N. Diaz, A. Naini, Y. Muthukumar, F. Sasse, M. Kalesse (2012) Synthesis of Simplified Tedanolide Analogues—Connecting Tedanolide to Myriaporone and Gephyronic AcidChemMedChem 2012, 7, 771
    DOI: 10.1002/cmdc.201100576
  • N. Diaz, M. Zhu, G. Ehrlich, U. Eggert, Y. Muthukumar, F. Sasse, M. Kalesse (2012) An Improved Route to (+)-Tedanolide and Analysis of Its Subtle Effects Controlling Conformation and Biological BehaviourChem. Eur. J. 2012, 18, 4946
    DOI: 10.1002/chem.201103038
  • O. Hartmann, M. Kalesse (2012) The Total Synthesis of (−)-Aurafuron AOrg. Lett. 2012, 14, 3064
    DOI: 10.1021/ol3011387
  • W. Zander, H. Irschik, H. Augustiniak, M. Herrmann, R. Jansen, H. Steinmetz, K. Gerth, W. Kessler, M. Kalesse, G. Höfle, R. Müller (2012) Sulfangolids, Macrolide Sulfate Esters from Sorangium cellulosumChem. Eur. J. 2012, 18, 6264
    DOI: 10.1002/chem.201100851
  • L. Bülow, A. Naini, J. Fohrer, M. Kalesse (2011) A Kiyooka Aldol Approach for the Synthesis of the C(14)–C(23) Segment of the Diastereomeric Analog of TedanolideOrg. Lett. 2011, 13, 6038
    DOI: 10.1021/ol202515x
  • M. T. Gieseler, M. Kalesse (2011) Asymmetric Vinylogous Mukaiyama Aldol Reaction of Aldehyde-Derived DienolatesOrg. Lett. 2011, 13, 2430
    DOI: 10.1021/ol2006727
  • A. Kena Diba, C. Noll, M. Richter, M. T. Gieseler, M. Kalesse (2010) Intramolecular Stereoselective Protonation of Aldehyde EnolatesAngew. Chem. Int. Ed. 2010, 49, 8367
    DOI: 10.1002/anie.201004619
  • B. Stauch, B. Simon, T. Basile, G. Schneider, N. P. Malek, M. Kalesse, T. Carlomagno (2010) Elucidation of the Structure and Intermolecular Interactions of a Reversible Cyclic-Peptide Inhibitor of the Proteasome by NMR Spectroscopy and Molecular ModelingAngew. Chem. Int. Ed. 2010, 23, 3934
    DOI: 10.1002/anie.201000140
  • D. Landsberg, M. Kalesse (2010) Synthesis of Symmetrical Ureas by (Diacetoxyiodo)benzene-Induced Hofmann RearrangementSynlett. 2010, 1104
    DOI: 10.1055/s-0029-1219566
  • I.E. Mohamed, S. Kehraus, A. Krick, G.M. Koenig, G Kelter, A Maier, H.H. Fiebig, M. Kalesse, N.P. Malek, H. Gross (2010) Mode of Action of Epoxyphomalins A and B and Characterization of Related Metabolites from the Marine-Derived Fungus Paraconiothyrium sp.J. Nat. Prod. 2010, 73, 2053
    DOI: 10.1021/np100310k
  • K. Rand; C. Noll; H. Martin Schiebel, D. Kemken; T. Dülcks, M. Kalesse, D. W. Heinz, G. Layer (2010) Oxygen-independent coproporphyrinogen III oxidase HemN utilizes harderoporphyrinogen as a reaction intermediate during conversion of coproporphyrinogen III into protoporphyrinogen IXBiol. Chem. 2010, 391, 55
    DOI: 10.1515/bc.2010.006
  • L. Bülow, I. Nickeleit, A.-K. Girbig, T. Brodmann, A. Rentsch, U. Eggert, F. Sasse, H. Steinmetz, R. Frank, T. Carlomagno, N. P. Malek, M. Kalesse (2010) Synthesis and Biological Characterization of Argyrin FChemMedChem. 2010, 5, 832
    DOI: 10.1002/cmdc.201000080
  • M. Cordes, M. Kalesse (2010) Heterocyclic and Acyclic Dienoxy Silane Synthons: Application in Total SynthesisChemTracks-Organic Chemistry 2010, 153
  • R. Schäckel, B. Hinkelmann, F. Sasse, M. Kalesse (2010) The synthesis of novel DisorazolesAngew. Chem. Int. Ed. 2010, 49, 1619
    DOI: 10.1002/anie.200906450
  • T. Brodmann, D. Janssen, F. Sasse, H. Irschik, R. Jansen, R. Müller, M. Kalesse (2010) Isolation and Synthesis of Chivotriene, a Chivosazole shunt Product from Sorangium cellulosumEur. J. Org. Chem. 2010, 5155
    DOI: 10.1002/ejoc.201000781
  • T. Brodmann, D. Janssen, M. Kalesse (2010) Total Synthesis of Chivosazol FJ. Am. Chem. Soc. 2010, 132, 13610
    DOI: 10.1021/ja107290s
  • T. Brodmann, N. D. Gomez, M. Kalesse (2010) Zwischen molekularem Werkzeug und medizinischer AnwendungNachr. Chem. 2010, 58, 131
    DOI: 10.1002/nadc.201069109
  • G. Hagelueken, S. C. Albrecht, H. Steinmetz, R. Jansen, D. W. Heinz, M. Kalesse, W.-D. Schubert (2009) The absolute configuration of rhizopodin, a potent inhibitor of actin polymerization, and its mode of actin dimerizationAngew. Chem. 2009, 121, 603
    DOI: 10.1002/ange.200802915
  • M. Lorenz, N. Bluhm, M. Kalesse (2009) Studies on the C22-C23 Aldol Coupling of SpirangienSynthesis 2009, 3061
    DOI: 10.1055/s-0029-1216918
  • S. Simsek, M. Kalesse (2009) Enantioselective synthesis of polyketides through vinylogous Mukaiyama aldol reactionsTetrahedron Lett. 2009, 50, 3485
    DOI: 10.1016/j.tetlet.2009.03.013
  • T. Brodmann, M. Lorenz, R. Schäckel, S. Simsek, M. Kalesse (2009) Highly Stereoselective Aldol Reactions in the Total Syntheses of Complex Natural ProductsSynlett 2009, 2, 174
    DOI: 10.1055/s-0028-1087520
  • G. Ehrlich, J. Hassfeld, U. Eggert, M. Kalesse (2008) The Total Synthesis of (+)-TedanolideJ. Am. Chem. Soc. 2006, 128, 14038
    DOI: 10.1021/ja0659572
  • G. Ehrlich, J. Hassfeld, U. Eggert, M. Kalesse (2008) The Total Synthesis of (+)-Tedanolide, a Macrocyclic Polyketide From Marine Sponge Tedania IgnisChem. Eur. J. 2008, 14, 2232
    DOI: 10.1002/chem.200701529
  • I. Nickeleit, S. Zender, F. Sasse, R. Geffers, G. Brandes, I. Sörensen, H. Steinmetz, S. Kubicka, J. Buer, A. Gossler, M. P. Manns, M. Kalesse, R. Frank, N. P. Malek (2008) Argyrin A - a p27kip1 stabilizing drug with potent antiproliferative and anti-angiogenic activityCancer Cell 2008, 14, 23
    DOI: 10.1016/j.ccr.2008.05.016
  • I. Nickeleit, S. Zender, F. Sasse, R. Geffers, G. Brandes, I. Sörensen, H. Steinmetz, S. Kubicka, T. Carlomagno, D. Menche, J. Buer, A. Gossler, M. P. Manns, M. Kalesse, R. Frank, N. P. Malek (2008) A myxobacterial cyclic peptide metabolite is a highly selective proteasome inhibitor and potent antitumor leadJournal of Peptide Science 2008, 14, 43
    DOI: 10.1002/psc.1089
  • M. Lorenz, M. Kalesse (2008) Synthesis of the C10-C32 Core Structure of Spirangien AOrg. Lett. 2008, 10, 4371
    DOI: 10.1021/ol8018105
  • M. Roy, M. Kalesse (2008) Synthesis of the TedanolidesNat. Prod. Rep. 2008, 25, 862
    DOI: 10.1039/B719607E
  • N. Schübel, M. Roy, M. Kalesse (2008) The Syntheses of the Tedanolides and MyriaporonesComptes Rendus Chimie 2008, 11, 1419
    DOI: 10.1016/j.crci.2008.05.013
  • U. Eggert, R. Diestel, F. Sasse, R. Jansen, B. Kunze, M. Kalesse (2008) Chondramide C: Synthesis, Configurational Assignment and First SAR StudiesAngew. Chem. Int. Ed. 2008, 47, 6478
    DOI: 10.1002/anie.200801156
  • D. Janssen, D. Abert, R. Jansen, R. Müller, M. Kalesse (2007) Chivosazole A – Elucidation of the full absolute and relative configurationAngew. Chem. Int. Ed. 2007, 46, 4898
    DOI: 10.1002/anie.200605198
  • D. Janssen, M. Kalesse (2007) Synthesis of the C15-C35 Segment of Chivosazole ASynlett 2007, 2667
    DOI: 10.1055/s-2007-991049
  • J. Liang, G. Ke, W. You, Z. Peng, J. Lan, M. Kalesse,A. M. Tartakoff, F. Kaplann T. Tao (2007) Interaction between importin 13 and myopodin suggests a nuclear import pathway for myopodinMolecular and Cellular Biochemistry 2008, 307, 93
    DOI: 10.1007/s11010-007-9588-1
  • M. Kalesse (2007) Aliphatic and Acyclic Aldehydes: Synthesis by ProtonationScience of Synthesis 2007, 25, 147
  • M. Kalesse (2007) Aliphatic and Acyclic Aldehydes: Synthesis by Elimination or RearrangementScience of Synthesis 2007, 25, 137
  • M. Kalesse (2007) Preface: Prof. Dr. Ekkehard WinterfeldtHeterocycles 2007, 74, 1
    DOI: 10.3987/COM-08-S(W)Preface_1
  • M. Lorenz, M. Kalesse (2007) Synthesis of the C23-C32 Fragment of SpirangienTet. Lett. 2007, 48, 2905
    DOI: 10.1016/j.tetlet.2007.02.081
  • N. Rahn, M. Kalesse (2007) The First Total Synthesis of ChlorotonilAngew. Chem. Int. Ed. 2008, 47, 597
    DOI: 10.1002/anie.200703930
  • S. Simsek. M. Horzella, M. Kalesse (2007) Oxazaborolidinone Promoted Vinylogous Mukaiyama Aldol ReactionsOrg. Lett. 2007, 9, 5637
    DOI: 10.1021/ol702640w
  • A. Stelmakh, T. Stellfeld, M. Kalesse (2006) Tandem Intramolecular Michael-Aldol Reaction as a Tool for the Construction of the C-Ring of Hexacyclinic AcidOrg. Lett. 2006, 8, 3485
    DOI: 10.1021/ol061096q
  • D. Ragunathan, V. M. Sanchez-Pedregal, J. Junker, M. Kalesse, A. Kirschning, T. Carlomagno (2006) TAR-RNA recognition by a novel aminoglycoside analogueNucl. Acid. Res. 2006, 34, 3599
    DOI: 10.1093/nar/gkl494
  • F. Liesener, M. Kalesse (2006) Synthesis of the C19-C26 Segment of AmphidinolideSynlett 2005, 2236
    DOI: 10.1055/s-2005-872236
  • F. Liesener, U. Jannsen, M. Kalesse (2006) Synthesis of a Northern Hemisphere of Amphidinolide H2Synthesis 2006, 2590
    DOI: 10.1055/s-2006-942459
  • G. Ehrlich, M. Kalesse (2005) Synthesis of the C13-C23 Segment of TedanolideSynlett 2005, 655
    DOI: 10.1055/s-2005-862391
  • M. Kalesse, J. Hassfeld, U. Eggert (2005) Synthesis of the C1-C17 Macrolactone of TedanolideSynthesis 2005, 1183
    DOI: 10.1055/s-2005-865302
  • N. Rahn, M. Kalesse (2005) A One-Pot Non-Aldol-Aldol Vinylogous Mukaiyama Aldol Tandem Sequence for the Rapid Construction of Polyketide FrameworksSynlett 2005, 863
    DOI: 10.1055/s-2005-863743
  • A. Kirschning, M. Lindner, M. Kalesse (2004) Synthesis of extended spacer-linked neooligodeoxysaccharides by metathesisolefination and evaluation of their RNA-binding propertiesTetrahedron 2004, 60, 3505
    DOI: 10.1016/j.tet.2004.02.013
  • B. Witzenbichler, M. Kalesse, S. Knüppel, H. P. Schultheiss (2004) Ratjadone is a potent inhibitor of coronary smooth muscle cell proliferation and induces cell differentiationCirculation 2004, 60, 3505.
  • T. Stellfeld, U. Bhatt, M. Kalesse (2004) Synthesis of the A,B,C-Ring System of Hexacyclinic AcidOrg. Lett. 2004, 6, 3889
    DOI: 10.1021/ol048720o
  • A. Burzlaff, M. Kalesse, C. Kasper, T. Scheper (2003) Multi parameter in vitro testing of ratjadone using flow cytometryAppl. Microbiol. Bitechnol 2003, 62, 174
    DOI: 10.1007/s00253-003-1300-0
  • B. Witzenbichler, M. Kalesse, S. Knüppel, H. P. Schultheiss (2003) Ratjadone is a potent inhibitor of vascular smooth muscle cell proliferationEuropean Heart Journal 2003, 24, 333
    DOI: 10.1016/S0195-668X(03)94882-2
  • M. Kalesse, M. Quitschalle, C.P. Khandavalli, A. Burzlaff, C. Kasper, T. Scheper (2003) The Total Synthesis of (−)‐Callystatin AChem. Eur. J. 2003, 9, 1129
    DOI: 10.1002/chem.200390130
  • J. Hassfeld, M. Kalesse (2002) Synthesis of the C1-C11 Segment of Tedanolide via Vinylogous Mukaiyama Aldol ReactionSynlett 2002, 12, 2007
    DOI: 10.1055/s-2002-35582
  • J. Hassfeld, M. Kalesse (2002) Advances in the vinylogous Mukaiyama aldol reaction and its application to the synthesis of the C1-C7 subunit of oleandolideTetrahedron Lett., 2002, 43, 5093
    DOI: 10.1016/S0040-4039(02)00993-0
  • M. Kalesse, M. Christmann (2002) The Chemistry and Biology of the Leptomycin familySynthesis 2002, 8, 981
    DOI: 10.1055/s-2002-31946
  • J. Hassfeld, M. Christmann and M. Kalesse (2001) Rapid access to polyketide scaffolds via vinylogous Mukaiyama aldol reactionsOrg. Lett. 2001, 3, 3561
    DOI: 10.1021/ol016677o
  • K. Michaelis, M. Kalesse (2001) Selective Cleavage of Unpaired Uridines with a Tyrosine-Cyclen ConjugateChemBioChem. 2001, 1, 79
    DOI: 10.1002/1439-7633(20010105)2:1<79::AID-CBIC79>3.0.CO;2-6
  • M. Christmann, M. Kalesse (2001) Vinylogous Mukaiyama Aldol Reactions with TriarylboranesTetrahedron Lett. 2001, 42, 1269
    DOI: 10.1016/S0040-4039(00)02254-1
  • M. Christmann, U. Bhatt, M. Quitschalle, E. Claus, M. Kalesse (2001) The Total Synthesis of (+)-RatjadoneJ. Org. Chem. 2001, 66, 1885
    DOI: 10.1021/jo005768g
  • M. Christmann, U. Bhatt, M. Quitschalle, Winfried Beil, Arne Burzlaff, Cornelia Kasper, L.-O. Haustedt, E. Hofer, T. Scheper, M. Kalesse (2001) The Biology and Chemistry of RatjadoneChemBioChem 2001, 2, 709
    DOI: 10.1002/1439-7633(20010903)2:9<709::AID-CBIC709>3.0.CO;2-7
  • M. Kalesse, M. Quitschalle, C.P. Khandavalli, A. Saeed (2001) Total Synthesis of (−)-Callystatin AOrg. Lett. 2001, 3, 3107
    DOI: 10.1021/ol016365l
  • M. Quitschalle, M. Christmann, U. Bhatt, M. Kalesse (2001) Synthesis of Unsaturated Lactone Moieties by Asymmetric Hetero Diels-Alder Reactions with Binaphthol-Titanium ComplexesTetrahedron Lett. 2001, 42, 1263
    DOI: 10.1016/S0040-4039(00)02213-9
  • M. Christmann, U. Bhatt, M. Quitschalle, E. Claus, M. Kalesse (2000) Total Synthesis of (+)-RatjadoneAngew. Chem. Int. Ed. 2000, 39, 4364
    DOI: 10.1002/1521-3773(20001201)39:23<4364::AID-ANIE4364>3.0.CO;2-G
  • M. Kalesse (2000) The Chemistry and Biology of DiscodermolideChemBioChem. 2000, 1, 171
    DOI: 10.1002/1439-7633(20001002)1:3<171::AID-CBIC171>3.0.CO;2-D
  • E. Claus, M. Kalesse (1999) Synthesis of the C6-C16 Polyene Fragment of Ratjadone, a Potent Cytotoxic Metabolite from Sorangium CellulosumTetrahedron Lett. 1999, 40, 4157
    DOI: 10.1016/S0040-4039(99)00716-9
  • K. Gerlach, M. Quitschalle, M. Kalesse (1999) Synthesis of the Northern Hemisphere of Epothilone A by a Ten-Membered Ring Closing Metathesis ReactionTetrahedron Lett. 1999, 40, 3553
    DOI: 10.1016/S0040-4039(99)00550-X
  • K. Michaelis, M. Kalesse (1999) Selective Cleavage of the HIV-1 TAR RNA with a Peptide-Cyclen ConjugateAngew. Chem. Int. Ed. 1999, 38, 2243
    DOI: 10.1002/(SICI)1521-3773(19990802)38:15<2243::AID-ANIE2243>3.0.CO;2-V
  • M. Kalesse, M. Quitschalle, E. Claus, K. Gerlach, A. Pahl, H.H. Meyer (1999) The Formal Total Synthesis of Epothilone AEur. J. Org. Chem. 1999, 2817
    DOI: 10.1002/(SICI)1099-0690(199911)1999:11<2817::AID-EJOC2817>3.0.CO;2-L
  • M. Quitschalle and M. Kalesse (1999) Improved Synthesis of the Northern Hemisphere of Epothilone A by a Sharpless Asymmetric DihydroxylationTetrahedron Lett., 1999, 40, 7765
    DOI: 10.1016/S0040-4039(99)01659-7
  • T. Oost, M. Kalesse (1999) Synthesis of Steroid Derived RNAse Active Site Model Systems: Modification of the C17 Pendant Imidazole and Substitution of the Guanidinium GroupsPolish. J. Chem. 1999, 73, 89
  • Tetrahedron Lett., 1999, 40, 7201 (1999) The Synthesis of the C15-C24 Segment of RatjadoneM. Christmann, M. Kalesse
    DOI: 10.1016/S0040-4039(99)01486-0
  • K. Gerlach, M. Quitschalle, M. Kalesse (1998) Synthesis of the C7-17 Segment of Epothilones by a 10-membered Ring Closing Metathesis ReactionSynlett 1998, 1108
    DOI: 10.1055/s-1998-1870
  • M. Kalesse, R. Wartchow (1998) Structural Features for the Promotion of Optimal Stacking in the Solid StateTetrahedron 1998, 54, 8015
    DOI: 10.1016/S0040-4020(98)00427-X
  • E. Claus, A. Pahl, P.G. Jones, H.H. Meyer, M. Kalesse (1997) Synthesis of the C1-C9 Segment of EpothilonsTetrahedron Lett. 1997, 38, 1359
    DOI: 10.1016/S0040-4039(96)02493-8
  • M. Kalesse (1997) Book Review: Organic and Bio-organic Mechanisms. By M. Page and A. WilliamsAngew. Chem. Int. Ed. 1997, 36, 2528
    DOI: 10.1002/anie.199725281
  • S. Mensching, M. Kalesse (1997) Generation of Thiazoles by Column Dehydrogenation of Thiazolidines with MnO2J. Prakt. Chem. 1997, 339, 96
    DOI: 10.1002/prac.19973390118
  • T. Oost, A. Filippazzi, M. Kalesse (1997) Bis(guanidinium) Receptors as Ribonuclease Active-Site Model Systems: Structural Changes and Solvent EffectsLiebigs Ann./Recueil 1997, 1005
    DOI: 10.1002/jlac.199719970532
  • T. Oost, M. Kalesse (1997) Synthesis of RNAse Active Site Model Systems Using a Steroid TemplateTetrahedron 1997, 53, 8421
    DOI: 10.1016/S0040-4020(97)00526-7
  • M. Kalesse, A. Loos (1996) Remarkable Hydrolysis of Phosphodiester by Neutral Lanthanide(III) DO3A ComplexesBioorganic & Medicinal Chemistry Letters 1996, 6, 2063
    DOI: 10.1016/0960-894X(96)00386-1
  • M. Kalesse, A. Loos (1996) Transesterification of Phosphodiester by a Zinc-Containing Cyclen Derivative: Identification of the Active SpeciesLiebigs Ann. 1996, 935
    DOI: 10.1002/jlac.199619960611
  • M. Kalesse, M. Eh (1996) Enantioselective Synthesis of the C1-C9 Segment of Bryostatin by Kinetic Resolution of Racemic β-Keto EstersTetrahedron Lett. 1996, 37, 1767
    DOI: 10.1016/0040-4039(96)00172-4
  • M. Kalesse, T. Wirth (1996) Bioorganische ChemieNachr. Chem. 1996, 44, 1178
    DOI: 10.1002/nadc.19960441212
  • M. Eh, D. Schomburg, K. Schicht, M. Kalesse (1995) An Efficient Synthesis of Radicinin AnaloguesTetrahedron 1995, 51, 8983
    DOI: 10.1016/0040-4020(95)00491-P
  • M. Eh, M. Kalesse (1995) Remarkable Kinetic Resolution of Chiral β-keto Esters by Baker-Yeast ReductionSynlett 1995, 837
    DOI: 10.1055/s-1995-5083
  • D. Schinzer, M. Kalesse (1991) Diastereoselective Double Michael Addition of Vinylogous Esters and Thexyldimethylsilyl Trifate-induced CyclizationsTetrahedron Lett. 1991, 32, 4691
    DOI: 10.1016/S0040-4039(00)92283-4
  • D. Schinzer, M. Kalesse (1989) Silica Gel-catalyzed Cyclization of Enones and Double Michael Additions of Vinylogous Amides: Efficient Synthesis of Bicyclo[2.2.2]octanones and Bicyclo-HydrocarbazolesSynlett 1989, 34
    DOI: 10.1055/s-1989-34704
  • D. Schinzer, M. Kalesse, J. Kabbara (1988) Silica Gel-catalyzed Cyclization of Mixed Ketene AcetalsTetrahedron Lett. 1988, 41, 5241
    DOI: 10.1016/S0040-4039(00)80726-1

Bücher

  • M. H. C. Cordes, M. Kalesse (2019) The Asymmetric Vinylogous Mukaiyama Aldol ReactionOrganic Reactions, Wiley
    DOI: 10.1002/0471264180.or098.02
  • L. Millbrodt, M. Kalesse (2017) Biology and Synthesis of the ArgyrinsCyclic Peptides, RSC Publishing, Cambridge, 2017, 122-140
    DOI: 10.1039/9781788010153-00122
    ISBN: 978-1-78262-528-5
  • F. Schaefers, T. A. M. Gulder, C. Bressy, M. Smietana, E. Benedetti, S. Arseniyadis, M. Kalesse, M. Cordes (2016) PolyketidesFrom Biosynthesis to Total Synthesis: Strategies and Tactics for Natural Products, John Wiley & Sons, Inc, Hoboken, NJ, 2016, 21-129
    DOI: 10.1002/9781118754085.ch2
    ISBN: 978-1-11875-173-2
  • M. Kalesse, A. Böhm, A. Kipper, V. Wandelt (2016) Synthesis of AntibioticsHow to Overcome the Antibiotic Crisis, Springer, Cham. 2016, 419-445
    DOI: 10.1007/82_2016_502
    ISBN: 978-3-319-49282-7
  • M. Kalesse (2014) In Silico Models for Drug Discovery. Edited by Sandhya KortagereChemMedChem. 2014, 9, 856
    DOI: 10.1002/cmdc.201400063
    ISBN: 978‐1‐62703‐341‐1
  • M. Cordes, M. Kalesse (2013) The vinylogous Mukaiyama aldol reaction in natural product synthesisModern Methods in Stereoselective Aldol Reactions, Wiley-VCH, Weinheim, 2013, 83-154
    DOI: 10.1002/9783527656714.ch2
    ISBN: 9783527332052
  • M. Kalesse, J. Hassfeld (2008) Asymmetric Vinylogous Mukaiyama Aldol ReactionAsymmetric Synthesis – The Essentials (2nd Edition), Wiley-VCH, Weinheim, 2008, 112-116
    ISBN: 978-3-527-32093-6
  • M. Kalesse, J. Hassfeld (2007) Asymmetric Vinylogous Mukaiyama Aldol ReactionAsymmetric Synthesis – The Essentials, Wiley-VCH, Weinheim, 2007, 105-107
  • M. Kalesse, T. Oost (1999) RNAse active site model systemsBioorganic Chemistry, Wiley-VCH, Weinheim, 1999, 272-280

Patente

  • D. Manstein, M. Preller, M. Furch, M. Kalesse, N. Diaz (2012) Preparation of biphenyl compounds useful in the treatment of malaria and other parasitic disorders, Patent angemeldet (WO, Nr.: 2013/034756 A1)
  • D. Manstein, M. Preller, M. Kalesse (2012) Novel means and methods for treating malaria and other parasitic disorders, Patent angemeldet (EP, 2 727 911 A1)
  • M. Kalesse, U. Eggert (2012) Method For Producing Intermediates For The Production Of Macrocycles That Are Inhibitors Of The Proteasomic Degradation of P27, Such As Argyrin And Derivatives Thereof, Patent angemeldet (US, 20120295941 A1)
  • M. Kalesse, U. Eggert (2010) Improved method for preparing protected tryptophan derivatives for the production of macrocycles that are inhibitors of the proteasomic degradation of p27, such as argyrin and derivatives thereof, Patent angemeldet (WO, 2011/073173 A1)
  • M. Kalesse, L. Bülow, A. Rentsch, A.-K. Girbig, U. Eggert, N. Malek, R. Frank, T. Brodmann (2009) Method for Producing Intermediates for the Production of Novel Macrocycles that are Inhibitors of the Proteasomic Degradation of p27, such as Argyrin and Derivatives Thereof, and Uses of Said Macrocycles, Patent angemeldet (US, 20110311564 A1)
  • M. Kalesse, N. Malek, R. Frank, T. Brodmann, L. Bülow, A. Rentsch, A.-K. Girbig, U. Eggert (2009) Method for producing intermediates for the production of novel macrocycles that are inhibitors of the proteasomic degradation of p27, such as argyrin and derivatives thereof, and uses of said macrocycles, Patent angemeldet (WO, 2010/006682 A1)
  • M. Kalesse, N. Malek, R. Frank (2008) Method for producing intermediates for the production of novel macrocycles that are inhibitors of the proteasomic degradation of p27, such as argyrin and derivatives thereof, and uses of said macrocycles, Patent angemeldet (EP, 2 138 507 A1)
  • U. Bhatt, C. P. Khandavalli, M. Christmann, M. Quitschalle, T. Scheper, W. Beil, A. Burzlaff, C. Kasper, E. Claus, M. Kalesse (2001) Ratjadon-Derivate zum Hemmen des Zellwachstums, Patent angemeldet; (DE, Nr.: 100 47 794.1)